Movoglechen ke motsoako oa bobeli oa sulfonylurea o nang le phello ea hypoglycemic 'meleng. Mochine oa ts'ebetso o ipapisitse le ho eketsa kutloelo-bohloko ea lisele tsa mmele ho insulin le ho matlafatseng sechertion ea lihormone ea lisele tsa pancreatic beta. Ts'ebetsong ea bongaka, sethethefatsi sa hypoglycemic se fuoe mofuta oa lefu la tsoekere la 2. Ha hoa lumelloa ho sebelisoa le lefu la tsoekere le itšetlehileng ka insulin.
Lebitso la Machaba le sa Tšoanelehang
Glipizide. Ka Latin - Glipizide.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu.png)
Motsamaisi oa lithethefatsi Movoglecen o na le lebitso la machaba la tlhaho e le Glipizide.
ATX
A10BB07.
Lokolla liforomo le sebopeho
Moriana o etsoa ka mokhoa oa litekanyetso tsa matlapa a tšoeu. Ka lehlakoreng le ka pele la yuniti ea lithethefatsi, ho na le kotsi e betliloeng, ha mongolo oa lengolo "U" moleng o bonahala o hlaha morao. Foromo ea Letlapa le le leng e na le 5 mg ea motsoako o sebetsang - glipizide. Ho eketsa sekhahla sa ho monya le bioavailability, konokono ea letlapa e na le likarolo tse ling:
- setlolo sa pregelatinized;
- hypromellose;
- tsoekere ea lebese;
- stearic acid;
- microcrystalline cellulose.
Matlapa a na le sebopeho se chitja sa cylindrical, se koahetsoe mothating oa ho qetela oa tlhahiso ke filimi ea enteric. Qetellong e na le talc, titanium dioxide, macrogol. Litsi tsa meriana li kenngoa ka har'a lithutsoana tsa lithutsoana tse 24. Ka lebokoseng la lebokose ho behiloe matlapa a 48.
Ketso ea pharmacological
Motsoako o tsoang ho hypoglycemic o tsoang ka molomong ke sulfonylurea.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu.jpg)
Movoglechen ea lithethefatsi e ama ts'ebetso ea manyeme mme ka nako e ts'oanang e na le phello e ntle ea "pancreatic".
Sehlahisoa se kopantsoeng ke sa moloko oa II. Mochine oa ts'ebetso oa karolo e sebetsang o ama ts'ebetso ea makhopho mme ka nako e ts'oanang o na le phello e eketsehileng-pancreatic. Glipizide e etsa hore ts'ebetso ea tlhahiso ea "insulin" e hlahisoe ke lisele tsa "pancreatic beta" nakong ea ho ts'oaroa ke lithane ka tsoekere, e matlafatse ts'ebetso ea lisele tsa kahare ho phello ea lihormone.
Ts'ebetsong ea ho fihlela phello ea kalafo, k'hemik'hale e sebetsang e eketsa monyetla oa ho tlama insulin ho lisa lisele, ho eketsa ho lokolloa ha hormone ea pancreatic. Ka lebaka leo, phello ea inulin ea insulin ho limolek'hule tsa tsoekere e ea matlafatsoa, 'me tekanyo ea ho monya tsoekere ka mesifa ea marapo le hepatocytes ea eketseha. Ho na le ho fokotseha ha gluconeogenesis ho sebete le ho phatloha ha lipid ho tishu ea adipose.
Botebo ba phello ea kalafo bo itšetlehile ka palo ea lisele tse sebetsang tsa beta ea manyeme.
Ka moriana lithethefatsi li na le phello e fokotsang fibrinolytic, diuretic le lipid-inhibits, 'me li lateloa ke ho etsoa ha sehokelo sa mali.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu.jpeg)
Movoglechen inhibits adhesion ea mokokotlo, e lateloe ke sebopeho sa thrombus.
Mofumahali
Kamora ho sebelisoa, moemeli oa "hypoglycemic" o haufi le ho kenella ka botlalo ka leboteng la mala a manyane a proximal ka lebelo le phahameng.
Ho ja lijo ka nako e tšoanang ha ho bake liphetoho lipakeng tsa litekanyetso tsa pharmacokinetic. Maemong ana, nako ea ho monya e eketseha ka metsotso e 45. Ha moriana o kenngoa tsamaisong ea methapo, lipalo tse phahameng tsa plasma li ka beoa nakong ea lihora tse 1-3 kamora ho sebelisa letlapa le le leng.
Bioavailability ea glipizide e fihla ho 90%. Maling, karolo e sebetsang e tlama albin ka 98-99%. Ha glipizide e feta li-hepatocytes, ntho e sebetsang e manehiloe lihlahisoa tsa metabolic tse sa bontsheng ts'ebetso ea hypoglycemic. Ho felisoa ha halofo ea bophelo ho etsa lihora tse 2-4. Setlhare sena se qhekelloa ka 90% ka sebopeho sa metabolites ka liphio, 10% ka sebopeho sa eona sa pele.
Matšoao a ho sebelisoa
Matlapa a Movoglechen a ka fokotsa khatello ea plasma ea tsoekere ea mofuta oa 2 lefu la tsoekere haeba lefu la tsoekere le sa itšetleheng ka insulin le sa phekoloe ka kalafo ea ho ja, boikoetliso le mehato e meng ea ho fokotsa boima bo feteletseng.
Contraindication
Ho nka meriana ho thibetsoe maemong a latelang:
- ho tsebahala ha methapo ea lisele ho sulfonamides, glipizide, likarolo tse ling tsa Movogleken kapa li-sulfonylurea;
- mofuta oa 1 lefu la tsoekere;
- lefutso la lefutso la tsoalo, lefu la tsoekere le lefu la galactose, ho haella ha lactase;
- ho chesa le ho kenella ha ts'ebetso ea sebaka se pharaletseng sa ts'ebetso, maemo a bohloko a morao-rao le likotsi, lits'ebetso tsa tšoaetso le ho ruruha;
- lefu la tsoekere le hyperosmolar coma, boemo bo botle;
- ketoacidosis;
- mafu a matla a sebete le a liphio.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-2.jpg)
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-2.jpeg)
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-3.jpg)
Hoa hlokahala ho fana ka litlhare ka ho lekola ka hloko boemo ba matšoao a bang teng ha motho a e-na le bothata ba ho ikhula.
Mokhoa oa ho nka Movoglechen
Litekanyetso li fetoloa ke ngaka ho latela boima ba 'mele le lilemo tsa mokuli, hammoho le litšobotsi tsa ts'ebetso ea methapo ea methapo.
Ngaka e ka etsa liphetoho ho regimen ea dosing ka liphetoho tse matla maemong a tsoekere ea serum.
Ka hona, ho hlahlojoa ka hloko ha tsoekere ea mali ho hlokahala: matšoao ka mpeng e se nang letho le ka mor'a lihora tse peli ka mor'a ho ja.
Le lefu la tsoekere
Matlapa a hlokahala bakeng sa tsamaiso ea molomo ka metsotso e 30 pele ho lijo. Hoseng pele ho lijo tsa hoseng, o lokela ho nka 5 mg ea moriana, ho sa sebetse letho kalafo, eketsa litekanyetso ka 2,5-5 mg, ho ipapisitse le mamello.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-4.jpeg)
Tekanyetso e kholo ea letsatsi le letsatsi ea Movoglek e lekaneng ke 40 mg, litekanyetso tsa ts'ebeliso e le 'ngoe ke 15 mg.
Sekhahla se phahameng se lumelletsoeng letsatsi ka leng ke 40 mg, litekanyetso tsa ts'ebeliso e le 'ngoe ke 15 mg. Matlapa a lokela ho tahoa 1 nako ka letsatsi. Ka tloaelo ea letsatsi le letsatsi e kaholimo ho 15 mg, ho hlokahala hore o arole litekanyetso ka litekanyetso tse 2,4.
Litla-morao tsa Movoglyken
Lisebelisoa tse hlophisitsoeng tse pepesang litlamorao tse mpe tsa lithethefatsi | Litlamorao tse mpe |
Sistimi ea Endocrine |
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Phekolo ea lijo |
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Ts'ebetso ea methapo le litho tsa kutlo |
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Hematopoietic litho tsa ka hare |
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Letlalo le maikutlo a ho kula |
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Tse ling |
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Tšusumetso ho bokhoni ba taolo ea methapo
Sethethefatsi sa hypoglycemic ha se ame tsamaiso ea methapo le bokhoni bo botle ba koloi, kahoo nakong ea kalafo ha ho thibetsoe ho khanna koloi kapa ho sebetsa ka lisebelisoa tse rarahaneng tse hlokang karabelo e potlakileng le khatello ea maikutlo.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-6.jpg)
Nakong ea kalafo le Movogleken ha ho thibetsoe ho khanna koloi.
Litaelo tse khethehileng
Litekanyetso li ntlafatsoa ha ho e-na le maemo a sithabetsang a bakang tahlehelo ea taolo ea maikutlo le maikutlo, maemong a boima bo matla ba 'mele, ka phetoho ea lijo.
Ha o theola lefu la tsoekere le sa itšetleheng ka insulin ha o fana ka ts'ebetso ea ts'ebetso, ho bohlokoa ho buisana le ngaka ea hau mabapi le kalafo e nchafalitsoeng ke insulin.
Pele a fana ka motsoako oa hypoglycemic, mokuli o lokela ho tsebisoa hore menyetla ea ho ba le hypoglycemia le lefu la tsoekere le eketseha ka joala, lithethefatsi tse seng khahlanong le ts'oaetso tsa mmele le ho tepella ka nako e telele. Ha o noella lino tse tahang, ho ka ba le karohano e kang ea ho hloka toka, e nang le bohloko ba ka mpeng, ho hlatsa le ho nyekeloa hoa pelo.
Ho fokotsa kotsi ea hypoglycemia ka lebaka la mafu a tšoaetsanoang, lihlahisoa tsa bohloeki li tlameha ho sebelisoa ho thibela ena.
Ka tšebeliso ea nako e telele ea Movoglecen, hoa khonahala ho hanyetsa ketso ea moriana ka ho fokolisa phello ea kalafo e latelang. Tabeng ena, ho khothalletsoa ho eketsa litekanyetso tsa letsatsi le letsatsi tsa lithethefatsi kapa ho kenya moemeli oa hypoglycemic.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-7.jpg)
Moriana ona o thibetsoe bana ba ka tlase ho lilemo tse 18.
Mosebetsi ho bana
Moriana ona o thibetsoe bana ba ka tlase ho lilemo tse 18 ka lebaka la tlhaiso-leseling e mabapi le phello ea glipizide holima kholo le kholo ea 'mele oa motho bongoaneng le bohlankaneng.
Sebelisa nakong ea bokhachane le pelehi
Ha ho tsejoe hore na karolo ea lik'hemik'hale e sebetsang e ka ama ts'ebetso ea ntshetsopele ea embryonic joang. Ke khopolo ea ho kenella ea glipizide ka thello ea hematoplacental ka tlolo ea molao ea morao-rao ea bookmark ea musculoskeletal system. Mabapi le hypotheses tsena, basali ba baimana ba thibetsoe ho sebelisa lithethefatsi tsa hypoglycemic bakeng sa tsamaiso ea molomo.
Ho khothalletsoa ho sebelisa li-cartridge le insulin ea motho ho fokotsa maemo a tsoekere.
Nakong ea kalafo le Movogleken, ho bohlokoa ho fetisetsa ngoana phepelong ea phepo e nepahetseng le ho emisa ho anyesa.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-8.jpg)
Nakong ea kalafo le Movogleken, ho hlokahala ho fetisetsa ngoana phepelong ea phepo e nepahetseng.
Kopo ea ts'ebetso ea renal e senyehileng
Mafung a matla a liphio, ho sebelisa moriana ona ho thibetsoe ka thata, hobane moriana o hloekisoa ka har'a moroto.
Sebelisa bakeng sa ts'ebetso ea sebete e sa sebetseng
Hoa hlokahala ho laola ts'ebetso e sebetsang ea sebete le li-enzyme tsa eona ka bonolo ho isa tekanyong e lekaneng ea ho haella. Ha ho na le ts'ebetso e boletsoeng ea pathological, phekolo ea lithethefatsi e thibetsoe.
Tekanyetso e feteletseng ea Movoglyken
Ho sebelisa lithethefatsi hampe ho ka lebisa ho hypoglycemia. Boemo bo tsamaea le:
- boikutlo ba tlala e matla;
- ho feto-fetoha ha maikutlo ka tšohanyetso ho fetoha le ho hlonama le boemo bo mabifi;
- ho fufuleloa ho eketsehileng;
- ketsahalo ea boemo bo nyahamisang;
- ho hloka boroko;
- hypoglycemic coma;
- puo le bofokoli ba pono;
- ho tsepamisa maikutlo mohopolo;
- ho lahleheloa ke kelello.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-9.jpg)
Ho sebelisa sethethefatsi ka mokhoa o feteletseng ho ka baka mofufutso o eketsehileng.
Haeba mokuli a hlokomela, ho hlokahala ho mo fa tharollo ea tsoekere. Maemong a ho felloa ke matla a ho tseba, tharollo ea 40% ea dextrose e lokela ho tsamaisoa ka matla kapa lerotholi le lokela ho beoa ka tharollo ea glucose ea 5%. 1-2 mg ea glucagon e tsamaisoa ka tsela e sa sebetseng. Ha a folisa mmuso ha mokuli a hlaphoheloa, o lokela ho ja lijo tse nang le lik'habohaedreite tse ngata. Sena se hlokahala ho thibela nts'etsopele ea hypoglycemia. Ka lefu la mokokotlo, ho hlokahala kalafo ka Dexamethasone kapa Mannitol.
Ho sebelisana le lithethefatsi tse ling
Ho se lumellane ha pharmacological le miconazole ho bonoa.
E ntlafatsa phello ea hypoglycemic | Fokotsa phello ea kalafo ea litafole |
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![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-10.jpg)
Movoglecen e fokotsa phello ea kalafo ea furosemide.
Ho sebelisoa ka nako e tšoanang ha lithethefatsi tsa myelotoxic ho eketsa kotsi ea agranulocytosis, ho ka baka ponahalo ea thrombocytopenia.
Tekanyo ea joala
Ethyl joala bo ntlafatsa phello ea hypoglycemic, e sitisa tsamaiso ea hematopoietic, ho sebetsa ha sebete le ho eketsa monyetla oa ho koaloa ha mali ka lebaka la ho eketseha ha lisele tse khubelu tsa mali le liplatelete. Ethanol e ama tsamaiso ea methapo e kholo le trophism ea methapo ea kutlo, ka hona, hoa hlokahala ho tlohela tšebeliso ea joala bakeng sa nako ea kalafo le Movogleken.
Li-analog
U ka nka meriana ka e 'ngoe ea lithethefatsi tse latelang.
- Glenez;
- Glibenesis;
- Antidiab;
- Lefu la tsoekere.
Lipehelo tsa khefu ea khemisi
Moriana oa Hypoglycemic o rekisoa ka lengolo la ngaka.
A na nka reka ntle le lengolo la ngaka?
Ka lebaka la kotsi ea ho ba le komello ea hypoglycemic, ho thibetsoe ho sebelisa moriana o le mong ntle le likeletso tsa bongaka.
Theko ea Movoglechen
Theko e tloaelehileng 'marakeng oa litlama e fihla ho li-ruble tse 1,600.
Maemo a polokelo ea moriana
Ho khothalletsoa ho boloka matlapa a le sebakeng se arohaneng le pente ea UV ka mocheso oa + 8 ... + 25 ° C.
Letsatsi la ho felloa ke nako
Likhoeli tse 42.
![](http://img.diabetesentity.com/img/sayd-2020/1219/preparat-movogleken-instrukciya-po-primeneniyu-2.png)
Analogue ea Movogleken - sethethefatsi Diabeteson se bolokiloe sebakeng se ka thoko ho kenella ka UV.
Moqapi
Zhuhai United Laboratories Co, China.
Tlhahlobo ea Movogleken
Kristina Doronina, ea lilemo li 28, Vladivostok
Monna oa ka o na le tsoekere e phahameng ea mali. Ka lilemo tse 'maloa, ba ne ba sa fumane moemeli ea loketseng oa glycemic, hore ba se ke ba fokotsa tsoekere feela, empa le ho boloka litefiso ka har'a meeli e tloaelehileng. Nakong ea puisano e latelang, ho ile ha ngoloa matlapa a Movoglecen. Kamora matsatsi a 30 a kalafo, tsoekere e khutletse ho tloaelehileng, sethethefatsi se ile sa hlaha. Hona joale e ka hare ho 8,2 limilimithara, empa e molemo ho feta 13-15 mm, e neng e le teng pele.
Yaroslav Filatov, ea lilemo li 39, Tomsk
Moriana ha oa ka oa thusa qalong. Kamora ho sebelisa 5 mg hoseng, tsoekere e bolokiloeng kahare ho 10-13 mm, lekhopho la letlalo le ile la qala. Ka litekanyetso tse ntseng li eketseha ho fihlela 20 mg, tsoekere e ile ea fokotseha butle ka libeke tse peli ho isa ho 6 mm. Litla-morao li ile tsa itlela ka botsona. Empa pontšo ena e itšetlehile ka lijo le likhothaletso ho litaelo. Moriana o ke ke oa theola tsoekere ha o na le khaello ea phepo e nepahetseng.
Ulyana Guseeva, ea lilemo li 64, Krasnoyarsk
Ha a le lilemo li 62, tsoekere ea mali e ile ea nyolohela ho 8-10 mm. E qalile nakong ea selemo, kamora ho tlohela mosebetsi. O ile a qala ho phela bophelo ba ho lula fatše ka lebaka la ho hloka mosebetsi, e leng se ileng sa lebisa ho eketseha ha tsoekere maling. Gluconorm e kopaneng le Siofor ha li a lekana.Matlapa a hlalositsoeng a Movoglek. Tsoekere e fokotsehile ka makhetlo a 2. Ka tlase 8 mm ha e fokotsehe. Ha ke so bone litla-morao leha e le life bakeng sa lilemo tse peli. Ho fihlela hajoale o ntse a phela hantle, empa haeba e mpefala, ho tla ba molemo ho fetohela setlhareng se seng.