Setlhare se entsoeng Russia bakeng sa kalafo ea khatello e phahameng ea mali le lefu la pelo le sa foleng. Ketso e thehiloe ho vasodilation. Phello e tsitsitseng ea kliniki e hlaha libeke tse 2-3 kamora ho qala kalafo.
Lebitso la Machaba le sa Tšoanelehang
Hinapril. Lebitso la Latin ke Chinaprilum.
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Setlhare se entsoeng Russia bakeng sa kalafo ea khatello e phahameng ea mali le lefu la pelo le sa foleng.
ATX
C09AA06
Lokolla liforomo le sebopeho
E fumaneha ka mokhoa oa matlapa ka ho koahela filimi ka litekanyetso tsa 5,10, 20 kapa 40 mg ea ntho e sebetsang. Ho 1 blister - matlapa a 10. Lithutso li tletse ka lebokoseng la karete ea 3 likhomphutha.
Moetso oa letlapa o kenyelletsa ntho e sebetsang le lebitso le le leng la lithethefatsi (phofo e tšoeu, e qhibilihang ka metsing) le likarolo tse ling - likarolo tse tlamang, dae, thickener, jj.
Ketso ea pharmacological
Ketso ea lithethefatsi e ipapisitse le thepa ea quinapril ho thibela exopeptidase ebe ka tsela eo o fokotsa ho kopana ha lihormopeptide lihormone tse bakang vasoconstriction.
Ka lebaka la sena, methapo ea kutlo e atoloha, phepelo ea mali ho myocardium kamora hore ischemia e ntlafale, phallo ea mali methapong le methapo ea mokokotlo e eketseha, ho hanyetsa khatello ea maikutlo ho eketseha, palo ea li-arrhythmias tsa ventricular lia fokotseha, khatello ea mali le kotsi ea ho fokotseha ha "thrombosis" e fokotseha.
Mofumahali
Sekhahla sa ho fihla sehlohlolong se phahameng sa moriana maling ke hora e le 'ngoe ka mor'a ho tsamaisoa ka molomo. Ketso e tšoarella ho latela tekanyo e nkuoeng.
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Sekhahla sa ho fihla sehlohlolong se phahameng sa moriana maling ke hora e le 'ngoe ka mor'a ho tsamaisoa ka molomo.
Ho fufuleloa ka mpeng ho ka ba 60%, empa ho ka mpefatsoa ke ho ja lijo tse mafura haholo ka nako e le 'ngoe.
E theha metabolites ka har'a sebete, haholo-holo quinaprilat, e atamelaneng le liprotheine tsa plasma ka nako e fetang 90%.
E epolloa ka liphio le mala.
Matšoao a ho sebelisoa
E sebelisoa ka bobeli bakeng sa monotherapy hape e kopantsoe le mafu a kang:
- khatello ea methapo ea kutlo (sekheo sa mantlha, sa ntlafatso, se sa hlalosoang);
- ho nyekeloa ke pelo (diastolic, pelo, le dysfunction ea diastolic, rastidity rardidity, ho hloleha ha pelo).
Ka khatello ea khatello ea mali, ho tsamaisa ka nako e le 'ngoe ka li-diuretics tsa potasiamo le beta-blockers ho ka khoneha, mme ka ho nyekeloa ke pelo - ka pelo-beta-blockers, joalo-joalo.
Contraindication
Moriana o kopantsoe maemong a latelang:
- hyperreaction ho ntho e sebetsang kapa likarolo tse ling tsa letlapa;
- ho ima le ho nyekeloa ke mpa;
- bana le bacha (ho fihlela lilemo tse 18);
- ho ba teng ha nalane ea angioedema;
- lefu la tsoekere;
- mosebetsi o sa sebetseng oa renal;
- arterial hypotension;
- hyperkalemia
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Ho khethoa hoa khoneha, empa ka tlhokomeliso le ka tlasa taolo e sa khaotseng ea basebetsi ba bongaka haeba ho na le:
- kotsi ea methapo ea methapo;
- atherosclerosis ea maoto;
- mitral valve stenosis;
- cardiopathy e thibelang le liphetoho tsa hypertrophic;
- a lipeo tse fetisitsoeng;
- ho ferekana ha purine metabolism (gout);
- mafu a autoimmune systemic connective tiske;
- lefu la tsoekere;
- tlhokeho ea li-inhibitors tsa MTOR le DPP-4;
- mafu a hanyetsang a bronchopulmonary system a sa foleng.
Ho molemo ho qoba ho nka matlapa ana ho bakuli ba nang le lefu la sebete le tsoetseng pele e le ho qoba ho holofala ha hepatic coma.
Mokhoa oa ho nka quinapril?
Nka ka molomo, ho sa tsotelehe lijo. Letlapa le metsoa ntle le ho hlafuna, le hlatsuoa ka metsi a manyane.
Ka khatello ea mali, monoprint e ka etsahala, 'me hammoho le baemeli ba bang.
Tabeng ea monotherapy, kalafo e qala ka tekanyetso ea 10 mg hang mme butle-butle e eketseha ho 20 kapa 40 mg, ho latela katleho ea phello ea kliniki.
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Ka khatello ea mali, monoprint e ka etsahala, 'me hammoho le baemeli ba bang.
Motsoako o kopaneng le diuretics, ho tloha ho 5 mg ka letsatsi o behiloe hang ka keketseho ea matsatsi a latelang ho fihlela sephetho se lebelletsoeng se fihlella, empa eseng ho feta tekanyetso ea letsatsi le letsatsi e khothalletsoang.
Eketsa lethal dose hoo e ka bang hang ka khoeli. Palo e phahameng e lumelletsoeng ka letsatsi ha e sa feta 80 mg ea moriana.
Ho hloleha ha pelo ho hloka kalafo e kopaneng. Tabeng ena, moriana o qaloa ka makhetlo a 5 mg ka makhetlo a mabeli ka letsatsi, o lateloa ke keketseho ea maemo a mamello e sa feteng keketseho e le 'ngoe ka beke.
Ka ts'ebetso ea renal e sa sebetseng hantle, tekanyetso ea moriana e khethoa ho latela boemo ba tumello ea "creatinine" - lehoetla le phahameng haholoanyane. Hoa khoneha ho eketsa palo e nkang kliniki feela, botsitso ba lipalo tsa mali le ts'ebetso ea liphio.
Le lefu la tsoekere
Ho bakuli ba nang le lefu la tsoekere mellitus, ha ba sebelisa sethethefatsi sena sa antihypertensive, ho hlokahala hore ho be le tlhokomelo e sa feleng ea bongaka ka khetho ea tekanyetso e nepahetseng ea lithethefatsi tsa hypoglycemic le insulin, kaha phello ea bona e ntlafalitsoe.
Litla-morao tsa hinapril
Ho ka ba le litlamorao tse tsoang ho hematopoiesis, tsamaiso ea methapo e bohareng, litho tsa ho hema le ho ruruha, methapo ea methapo le pelo, letlalo, tseo hangata li sa buuoeng haholo. Bakeng sa linyeoe tse 100 tsa ho fana ka taelo, ke hoo e ka bang 6% feela ea linyeoe tsa ho tlosoa tse ngolisitsoeng.
Ka nako e 'ngoe ho na le tlolo ea phefumoloho le pono, ho fokotseha ha potency, bohloko mokokotlong le sefubeng, jj.
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Phekolo ea ka mpeng
Mohlomong ponahalo ea ho nyekeloa ke pelo, ho hlatsa, dyspepsia, pancreatitis, hepatic coma, necrosis ea sebete, angioedema ea mala.
Hematopoietic litho tsa ka hare
Anemia, thrombocytopenia, neutropenia, hyperkalemia, keketseho ea "metabolinine" e eketsehileng.
Tsamaiso ea methapo e bohareng
Ho opeloa ke hlooho khafetsa le ho tsekela. Ka linako tse ling paresthesia, khatello ea maikutlo le ho hloka boroko li etsahala.
Ho tsoa ts'ebetsong ea moroto
Ho hloleha ha renal haholo, ts'oaetso ea pampiri ea urine.
Karolong ea letlalo
Litla-morao li bontšoa ke pemphigus, baldness, ho fufuleloa ho eketsehileng, photosensitivity, le dermatitis.
Ho tsoa ho tsamaiso ea methapo ea pelo
Hypotension, failing, pherekano ea morethetho oa pelo, stroke, phomolo ea mabota a methapo ea mali.
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Allergie
Ho thothomela ha Anaphylactic le edema ea Quincke hoa khoneha.
Tšusumetso ho bokhoni ba taolo ea methapo
Ho hlokahala hore motho a be hlokolosi ha a khanna a bile a sebetsa, 'me a hloka hore motho a shebane haholo, hobane ka nako ea litla-morao a theohile haholo khatello ea mali le ho tsekela.
Litaelo tse khethehileng
Ka keketseho ea mocheso oa 'mele kapa tonsillitis, liteko tsa mali li lokela ho etsoa ho khetholla neutropenia.
Pele a etsa opereishene, ho kenyeletsa le meno, ngaka e tlameha ho lemosoa ka ho beoa ha chelete e hlalositsoeng pele.
Sebelisa botsofaling
Litšireletso li fanoa botsofaling ka lebaka la tekanyo e fokolisitsoeng ea ho tlosoa hoa eona 'meleng.
Mosebetsi ho bana
Ha e sebetse ho fihlela lilemo tse 18.
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Ka hloko, hinapril e beoa botsofaling ka lebaka la tekanyo e fokolitsoeng ea ho pepesa ha 'mele oa hau.
Sebelisa nakong ea bokhachane le pelehi
Nakong ea kemaro le ha ngoana a anyesa ngoana, tšebeliso ea li-inhibitors tsa ACE e thibetsoe ka thata. E na le bokhoni ba ho sitisa nts'etsopele le ho baka lefu la fetal. Nakong ea kanyeso, e ka fetela lebeseng mme ea baka karabelo e mpe ho lesea.
Bongata ba li-quinapril
Kamora ho nka tekanyo e fetang tekanyo e phahameng ea litekanyetso, ho senyeha ha pono, ho ka ba le khatello e matla ea maikutlo le ho ba le tsebiso. Phekolo ntlheng ena e fanoa ho latela matšoao.
Ho sebelisana le lithethefatsi tse ling
Ntlafatsa phello ea antihypertensive: li-analgesics tsa narcotic, litokisetso tsa khauta, anesthetics, diuretics, ACE inhibitors.
Fokotsa phello ea sodium chloride, li-estrogens, lithethefatsi tse seng khahlanong le ts'oaetso tsa mali.
E fokotsa ho amoheloa ha tetracycline.
Tabeng ea tšebeliso e le 'ngoe ka litokisetso tsa lithium, ho tahoa hoa lithium hoa khoneha.
E ntlafatsa ketso ea lithethefatsi tsa insulin le hypoglycemic.
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Hinapril e fokotsa ho amoheloa ha tetracycline.
Ha e khothalletsoe ho kopanya le Aliskiren, immunosuppressants, mTOR kapa DPP-4 enhibitors, hammoho le lithethefatsi tse thibelang ts'ebetso ea marapo.
Tekanyo ea joala
Joala bo ntlafatsa phello e matla ea khatello ea mali, ka hona, tšebeliso e kopantsoeng e kopantsoe.
Li-analog
Ka mokhoa o ts'oanang, matlapa a koahetsoeng ka filimi a sebetsa 'me a na le motsoako o tšoanang sebopeho:
- Accupro - 5.10, 20 kapa 40 mg (Jeremane).
- Akkuzid - 10 kapa 20 mg (Jeremane). Moriana o kopaneng. E na le ntho ea bobeli e sebetsang - hydrochlorothiazide.
- Hinapril C3 - 5.10, 20 kapa 40 mg (Russia).
- Quinafar - 10 mg (Hungary).
Matlapa a tšoanang sehlopheng sa litlhare:
- Amprilan - 1.25; 2,5; 5 le 10 mg (Slovenia).
- Vasolapril - 10 kapa 20 mg (Turkey).
- Diropress - 5, 10 kapa 20 mg (Slovenia).
- Captopril - 25 kapa 50 mg (Russia, India).
- Monopril - 20 mg (Poland).
- Perineva - 4 kapa 8 mg (Russia / Slovenia).
Li-Analog li ka ba tsa mekhahlelo e fapaneng ea theko.
Lipehelo tsa khefu ea khemisi
A na nka reka ntle le lengolo la ngaka?
E fanoa feela ka taelo ea ngaka ke ngaka e eang.
Theko ea Hinapril
Karolelano ea theko.
Boholo ba theko bo tsoa ho li-ruble tse 200 ho isa ho tse 250 ka sephutheloana, ho latela tekanyetso.
Maemo a polokelo ea moriana
Boloka mocheso oa kamoreng (e seng ho feta + 25ºC) sebakeng se lefifi, moo bana le liphoofolo tse ruuoang lapeng.
Letsatsi la ho felloa ke nako
Bophelo ba Shelf bakeng sa lilemo tse 3 ho tloha ka letsatsi la ho tsoa le ka mor'a letsatsi la ho felloa ke nako bo tlameha ho lahloa.
Moqapi
E etsoa Russia Russia k'hamphaning ea meriana ea Zoo Severnaya Zvezda.
Litlhahlobo tsa Hinapril
Lingaka
Irina, ngaka ea lelapa, Tver
Ke ngolla bakuli ba nang le khatello ea mali ea methapo ka mor'a ho bokella anamnesis le tlhahlobo e felletseng. Hangata ke kopanya le diuretics ho ea ka lipontšo. Setlhare se sebetsa hantle, empa o lokela ho lula o batla ka hloko boteng ba li-contraindication ho motho ka mong, hobane litla-morao tse kotsi li ka etsahala.
Sergey, ngaka ea methapo ea pelo, Astrakhan
Ka ho nyekeloa ke pelo, setlhare se joalo se fana ka liphallelo tse potlakileng, empa pele ho nako, u lokela ho etsa tlhahlobo le ho ithuta nalane ea bongaka.
Bakuli
Anna, ea lilemo li 52, Volgograd
Ke nooa lipilisi joalokaha ke laetsoe ke ngaka e le sesebelisoa se tšehetsang khatello ea mali. Ka litla-morao, ke khona ho bona ho otsela hanyane qalong ea kalafo.
Sophia, ea lilemo li 39, Vologda
Ho tloha khale haholo, mathata a khatello a ile a qala. Ke ile ho setsebi sa bongaka 'me moo, kamora tlhahlobo, lipilisi tsena li ile tsa beoa. Hona joale khatello e batla e le ntho e tloaelehileng, ntle le ha ho ba le merusu e matla, 'me ha ho kotuloe litholoana tse bosula tsa extraneous.