Mathata a vasulin a ka baka mafu a mangata. Phekolo ea bona e tla hloka kalafo e rarahaneng, e kenyelletsang ho sebelisa meriana, e kenyelletsang angiopril. Pele o sebelisoa, o hloka ho ithuta litaelo tse khothetsoeng ke moriana e le hore ho se be le mathata.
Lebitso la Machaba le sa Tšoanelehang
Lebitso la machaba le sa amehang bakeng sa sehlahisoa ke Captopril.
![](http://img.diabetesentity.com/img/sayd-2020/1289/preparat-angiopril-instrukciya-po-primeneniyu.jpg)
Bakeng sa kalafo ea bona ea methapo ea mali, kalafo e rarahaneng ea hlokahala, e kenyeletsang ho sebelisa meriana, e kenyeletsang angiopril.
ATX
Moriana o na le khoutu ea ATX e latelang: C09AA01.
Lokolla liforomo le sebopeho
Ho lokolloa ha moriana ho etsoa ka mokhoa oa matlapa a behiloeng ka mekhahlelo ea li-pcs tse 10 le likhomphutha tse 4. Letlapa la karete e ka ba le 1, 3, 10 strip ea matlapa a 10 e le 'ngoe kapa sekala se le seng se nang le matlapa a 4. Motsoako o sebetsang ke Captopril - 25 mg. Ntle le moo, ho sebelisoa li-stearic acid, lactose, starch ea poone, colloidal silicon dioxide le cellcose ea microcrystalline.
Ketso ea pharmacological
Ntho e sebetsang e thibela ts'ebetso ea enzyme e fetolang. E liehisa sebopeho sa angiotensin 1 le 2, e felisa phello ea eona ea vasoconstrictor methapong le methapong. Ho nwa moriana ho thusa ho fokotsa ho jarolla pele le kamora boima, khatello e tlase ea mali, ho fokotsa khatello ea methapo ea methapo, ho fokotsa ho tsoa ha aldosterone ka har'a litšoelesa tsa adrenal, le ho fokotsa khatello ea ho potoloha ha methapo ea mali le atrium e nepahetseng.
Mofumahali
Kamora ho nka matlapa, e kenella ka potlako pampiring ea mala ka lebaka la bioavailability ea 60-70%. Ho theoha butle butle ho bonoa ka tšebeliso ea nako e le 'ngoe ea lijo tsa batho ba bangata. Bophelo ba halofo ea lithethefatsi bo tla nka lihora tse 2-3. Hafu ea motsoako o sebetsang o tšeloa ka har'a moroto ka sebopeho se sa fetoheng.
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Matšoao a ho sebelisoa
Matšoao:
- khatello ea kelello ea methapo, ho kenyelletsa le ntlafatso ea kelello;
- lefu la tsoekere le lefu la tsoekere la mofuta oa 1;
- lefu la pelo le sa foleng;
- tšilafalo ea "ventricle" ea leqeleng kamora ho kenella ka har'a myocardial ho bakuli bao boemo ba bona ba kliniki bo tsitsitseng.
Contraindication
Basali baimana le ba robalang, bana ba ka tlase ho lilemo tse 18 le batho ba nang le mamello ho likarolo tsa lithethefatsi le li-inhibitors tse ling tsa ACE, hammoho le bakuli ba nang le lefu la mokokotlo oa cerebrovascular, ba lokela ho hana kalafo ka sethethefatsi.
U ka e nka joang
Setlhare se etselitsoe tsamaiso ea molomo. Matlapa a nooa makhetlo a 2-3 ka letsatsi ho 6.25-12.5 mg. Haeba ho hlokahala, palo ea meriana e eketsoa ho 25-50 mg. Tekanyo e phahameng ea letsatsi le letsatsi ha ea lokela ho feta 150 mg. Ha ho kgothaletswe ho fetola tekanyetso ka boyena.
Le lefu la tsoekere
Haeba mokuli a e-na le lefu la tsoekere, hona moriana o nooa ho 75-150 mg ka letsatsi. Litekanyetso li ka fetoloa ke mofani oa hau oa tlhokomelo ea bophelo.
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Haeba mokuli a e-na le lefu la tsoekere, hona moriana o nooa ho 75-150 mg ka letsatsi.
Litlamorao
Maemong a mang, karabelo e mpe ea 'mele ho tsoa tsamaisong ea methapo le litho tse ling li ka hlaha ka tsela ea:
- tachycardia;
- ho fokotsa khatello ea mali;
- edema ea peripheral;
- orthostatic hypotension;
- angioedema ea maoto, matsoho, li-membrane tsa mucous, sefahleho, larynx, leleme, molomo le pharynx;
- khohlela e omileng;
- pulmonary edema;
- bronchospasm;
- Ho tsekela
- hlooho e opang;
- ho senyeha ha pono;
- ataxia
- ho otsela
- paresthesia;
- thrombocytopenia;
- phokolo ea mali
- neutropenia;
- agranulocytosis;
- acidosis;
- proteinuria;
- hyperkalemia
- hyponatremia;
- maemo a eketsehang a "nitinine" le "nitrogen" ea mali maling;
- molomo o omileng;
- stomatitis;
- bohloko bo ka mpeng;
- likotsi tsa tatso;
- ho felloa ke takatso ea lijo;
- mosebetsi o eketsehileng oa li-enzyme tsa sebete;
- hyperbilirubinemia;
- hepatitis;
- lets'ollo
- gingival hyperplasia.
Haeba litla-morao li hlaha, matlapa a lokela ho emisoa.
Tšusumetso ho bokhoni ba taolo ea methapo
Bakuli ba noang sethethefatsi sena ba lokela ho ba hlokolosi ha ba khanna le ho etsa lintho tse hlokang ho tsepamisa maikutlo le ho ts'oarana le maikutlo ka potlako, ka lebaka la ponahalo ea ho tsofala.
Litaelo tse khethehileng
Nakong ea phekolo ea Angiopril, litholoana tse mpe tse fosahetseng li ka bonoa ka boitšoaro ba tlhahlobo ea moroto bakeng sa acetone. Ka hypotension ea arterial, palo ea lithethefatsi ea fokotseha. - Noa litafole ka hloko ka granulocytopenia.
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Ka hypotension ea arterial, palo ea lithethefatsi ea fokotseha.
Mosebetsi ho bana
Tšebeliso ea lithethefatsi ho phekola bana e thibetsoe. Pheko e ka khethoa maemong a khatello e matla ea mali. Pilisi e baloa ho latela boima ba ngoana. Ke 0,0-0.4 mg ea moriana ka kilo e le 'ngoe ea boima ba' mele. Ho amoheloa hangata ha hoa lokela ho feta makhetlo a mabeli ka letsatsi.
Sebelisa nakong ea bokhachane le pelehi
Ha u nkile ngoana le ho anyesa, li-captopril ha lia lokela ho tšoaroa. Haeba ho ima ho fumanoa ka nako ea kalafo, ho hlokahala ho emisa ho nka matlapa. Ha ho hlokahala, tsamaisa litekanyetso tsa kalafo tse anyesang.
Kopo ea ts'ebetso ea renal e senyehileng
Tabeng ea ho senyeha ha renal le ho se sebetse hantle ha masapo, ho hlokahala hore ho fokotsoe tekanyetso ea letsatsi le letsatsi.
Sebelisa bakeng sa ts'ebetso ea sebete e sa sebetseng
Ka hloko le ka tlasa taolo ea bongaka, ba sebelisa lithethefatsi bakeng sa mathata a sebete.
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Bongata
Haeba o sebelisa hampe meriana e khothalletsoang, ho ka 'na ha e-ba le mokhoa o mongata oa ho sebelisa lithethefatsi ka mokhoa oa ho fokotseha ka sekhahla ha khatello ea mali. Maemong ana, mokuli o kenngoa ka tharollo ea isotonic sodium chloride kapa mofuta o mong o nkang metsi a tsoang plasma le hemodialysis o etsoa.
Ho sebelisana le lithethefatsi tse ling
Ts'ebeliso e kopaneng ea indomethacin le lithethefatsi tse ling tse sa ts'oeng mali tsa antiidal li ka fokotsa phello ea hypotensive ea angiopril. Kotsi ea hyperkalemia e eketseha ka tšebeliso e ts'oanang ka lisebelisoa tse nang le letsoai, li-diuretics tse nang le potasiamo, litokisetso tsa potasiamo le tlatsetso ea potasiamo. Matla a antihypertensive a fokotsehile ka tšebeliso ea li-erythropoietins le acetylsalicylic acid.
Keketseho ea khatello ea serum ea lithium e ka bonoa ha e sebelisana le letsoai la lithium. Ho matlafatsa ts'ebetso ea moriana ho etsahala ha ho kopantsoe le diuretics le vasodilators. Mathata a amanang le lefu la kelello a ka hlaha ka ts'ebeliso e kopaneng ea li-antidepressants le Captopril. Bakuli ba sebelisang procainamide kapa allopurinol ba na le kotsi e eketsehileng ea neutropenia.
Tekanyo ea joala
Nakong ea kalafo, ho thibetsoe ho noa lino tse tahang. Ho sebelisana ha bona le karolo e sebetsang ho ka baka khatello e matla ea khatello ea mali.
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Nakong ea kalafo, ho thibetsoe ho noa lino tse tahang.
Li-analog
Haeba ho hlokahala, moriana o nkeloa sebaka ke analog. Har'a tsona ho na le tse latelang:
- Alkadil;
- Blockordil;
- Kapoten;
- Catopil;
- Epsitron.
Liphetoho kalafong li lokela ho etsoa ke ngaka e khethang lithethefatsi li nahanela litšobotsi tsa 'mele oa mokuli le ho teba ha methapo ea methapo.
Maemo a phomolo Angiopril a tsoang litlolong tsa litlama
Sesebelisoa se ka rekoa k'hemisteng ka taelo ea ngaka ho ngaka.
A na nka reka ntle le lengolo la ngaka?
Matlapa a ke ke a rekoa ntle le lengolo la ngaka.
Theko
Litsenyehelo tsa moriana li ipapisitse le leano la litheko tsa k'hemiste 'me ka kakaretso ke li-ruble tse 95.
Maemo a polokelo ea moriana
Setlhare se beoa sebakeng se lefifi, se omileng le se sa fumaneheng bakeng sa bana se nang le mocheso o sa feteng 25 ° C.
Letsatsi la ho felloa ke nako
Setlhare se boloka thepa ea sona ka lilemo tse 3 ho tloha ka letsatsi la tlhahiso, ho latela maemo a polokelo. Ha letsatsi la ho felloa ke nako le felletse, le tla lahloa.
Mohlahisi Angiopril
Sehlahisoa se hlahisa TORRENT PHARMACEUTICALS Ltd. (India).
![](http://img.diabetesentity.com/img/sayd-2020/1289/preparat-angiopril-instrukciya-po-primeneniyu-27.jpg)
Sesebelisoa se ka rekoa k'hemisteng ka taelo ea ngaka ho ngaka.
Litlhahlobo mabapi le Angiopril
Vladimir, ea lilemo li 44, Krasnoyarsk: "Ke sebelisitse lithethefatsi kamora ho kenella ka mpeng. Leha ho bile le litlamorao tse ngata, kalafo e tsamaile hantle. Ke hlophisitse theko ea Angiopril. E theko e tlase ebile e ea sebetsa. Ke e khothaletsa."
Larisa, ea lilemo li 24, Murmansk o re: "Ngaka e ile ea fana ka pheko ea lefu la tsoekere. O ile a nka chelete e nyane hoo e ka bang khoeli. Matsatsing a pele, ho ts'oaroa ke sefuba le khohlela e omileng li ile tsa nkhathatsa, empa nakong e tlang tsohle ha li a ka tsa fumana lithethefatsi hanghang, mme theko e ile ea makatsa. Ke ne ke nahana hore e theko e phahameng. kalafo e tla bitsa. "