Aprovel 300 ke lithethefatsi tse sebetsang tsa antihypertensive tsa moloko o mocha. E etselitsoe phekolo ea khatello ea methapo ea mali le ho thibela mathata a eona. Ka tšebeliso e nepahetseng le litekanyetso, litla-morao ha li shebelloe, katleho ea kalafo e fihlella kapele.
Lebitso la Machaba le sa Tšoanelehang
INN - Irbesartan.
ATX
C09CA04. E bolela ho thaepa II angiotensin receptor antagonists.
Lokolla liforomo le sebopeho
Sebopeho sa tlhahiso - matlapa a 150 kapa 300 mg. Sesebelisoa se sebetsang ke irbesartan. Ho feta moo, sebopeho sa matlapa a kenyelletsa lintho tse thusang ho monya motsoako oa lithethefatsi le ho thibela ho tenoa, ho senngoa ha letlapa.
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Sebopeho sa tlhahiso ke litafole, ntle le moo, sebopeho se kenyelletsa lintho tse thusang ho monya le ho thibela ho hoholeha, ho senngoa ha letlapa.
Ketso ea pharmacological
Lithethefatsi ke mohanyetsi oa li-receptor tsa angiotensin-2, ts'ebetso ea eona ke karolo ea bohlokoa ea pathogenetic ho khatello ea mali. Mori o thibela litlamorao tsohle tsa angiotensin, ha o na mosebetsi ho li-receptors tsa AT-1. Ha e ame ACE le renin, liteishene tsa ion tse kenyelletsoang ho boloka sostost homeostasis le ho laola khatello ea mali.
Ho nka moriana ka litlolo tse hlalositsoeng ka mokhoa o hlakileng ho fokotsa khatello ea aldosterone ho plasma, ha potasiamo e ntse e sa fetohe. Ho fokotseha ha khatello ho bonoa kamora tšebeliso ea eona ea pele mme e bonahala kamora beke. Lithuto tsa kliniki li tiisa ho bolokoa hoa phello ea nako e telele ea lithethefatsi.
Ka tekanyo e le 'ngoe ea ho fihlela ho 300 mg, ho fokotseha ha khatello ea mali ka 10/7 mm (ka karolelano) ho bonoa. Ha o sebelisa placebo, phello e nepahetseng ha e bonoe. Maemong a sa tloaelehang, ntshetsopele ea orthostatic e khonahala. Ho bakuli ba nang le sodium e khutsitseng maling, ho fokotseha ho feteletseng ha khatello hoa khoneha.
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Aprovel 300 ke lithethefatsi tse sebetsang tsa antihypertensive tsa moloko o mocha.
Ho sebetsa ha sethethefatsi ha hoa itšetleha ka lilemo kapa bong ba mokuli. Bathong ba morabe oa Negroid, phello ea meriana ha e hlahisoe. Kamora ho hlakoloa ha Aprovel, khatello e khutlela butle butle litekanyetsong tsa eona tsa pele.
Mofumahali
Kamora ho tsamaisoa ka molomo, moriana o kenella ka potlako maling. Bioavailability e nyolohetse ho 80%. Ts'ebetso e kholo ea plasma e fihlella ka mor'a lihora tse peli.
Metabolism e etsahala ka har'a sebete. Butle-butle li-metabolism li tsoa le liphio, bile, makhopho. Ha e fetohe, tekanyo e nyane haholo ea lithethefatsi e ea tlosoa. Nako eo ka eona e felisoang halofo ea 'mele e pakeng tsa lihora tse 11 ho isa ho tse 15.
Matšoao a ho sebelisoa
Moriana ona o khothalletsoa hore o sebelisoe maemong a latelang.
- khatello ea mali ea methapo (e le monotherapy hape e kopantsoe le lithethefatsi tse ling tsa antihypertensive);
- nephropathy e bakoang ke khatello ea mali le lefu la tsoekere la mofuta oa 2.
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Moriana ona o khothalletsoa hore o sebelisoe nakong ea khatello ea methapo ea methapo (e le monotherapy hape o kopantsoe le lithethefatsi tse ling tsa antihypertensive).
Contraindication
Moriana o kopantsoe maemong a latelang:
- sensitivity ho ntho e sebetsang kapa ntho efe kapa efe;
- kamohelo e le 'ngoe ea chelete ka Aliskiren;
- tšebeliso e kopanetsoeng ea li-inhibitors tsa ACE boteng ba lefu la tsoekere ho lephoka;
- lefutso le ikemiselitseng ho amohela galactose, lactase;
- ho hloleha ho matla ha sebete;
- nako ea boitšisinyo kapa nako ea ho anyesa;
- lilemo tsa bana.
Ka tlhokomelo
Tlhokomeliso e eketsehileng e lokela ho bonoa ho mafu le maemo a latelang:
- ho fokotsa li-valve tsa mitral kapa aortic;
- kalafo ea diuretic;
- fokotseha ha molumo oa mali o potoloha, o theohe maemong a sodium;
- cardiomyopathy;
- letsoai le lekanyelitsoeng;
- ho hlatsa
- mosebetsi o sa sebetseng oa renal;
- IHD, atherosclerosis ea lijana tse fepang boko;
- tšebeliso ea lithethefatsi tse seng khahlanong le ts'oaetso tsa steroidal (ho na le kotsi e eketsehileng ea ho hloleha ha liphio).
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Ho lebisoa tlhokomelo e eketsehileng ho lokela ho bonoa haeba ho na le mathata a ho sebetsa a renal.
Mokhoa oa ho nka Aprovel 300
Moriana o nooa feela ka molomo. Letlapa le metsoa kaofela 'me le hlatsuoa ka metsi a mangata. Nka hanngoe ka letsatsi hoseng pele u ja.
Le lefu la tsoekere
Ho lefu la tsoekere, ha ho na lebaka la ho fetola tekanyetso. Moriana o fanoa e le karolo ea kalafo e rarahaneng ho bakuli ba nang le lefu la tsoekere. Nakong ea kalafo, o lokela ho lula a lekola glucometer.
Litlamorao tsa Aprovel 300
Ha u sebelisa lithethefatsi, ponahalo ea litlamorao tse sa rateheng ea khoneha.
Phekolo ea ka mpeng
Khafetsa, bakuli ba ka ba le ho nyekeloa ke pelo, e tsamaeang le ho hlatsa, nako le nako - lets'ollo kapa ho sokela. Ho na le monyetla oa ho ba le mofuthu oa pelo.
Tsamaiso ea methapo e bohareng
Nakong ea kalafo le Aprovel, ho tsekela le ho opeloa ke hlooho ho ka hlaha. Nako le nako, boemo ba syncopal bo khonahala ka phetoho ea boemo ba 'mele. Ka linako tse ling ho senya litho tsa kutlo.
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Ho tsoa tsamaisong ea phefumoloho
Nako le nako, ho khohlela ho tšoenya bakuli.
Ho tsoa ts'ebetsong ea genitourinary
Mohlomong nts'etsopele ea khatello ea kelello ho banna.
Ho tsoa ho tsamaiso ea methapo ea pelo
Maemong a sa tloaelehang, nts'etsopele ea edema, ho eketseha ha sekhahla sa pelo hoa khoneha. Ka linako tse ling bakuli ba tšoenyeha ka mokhathala o akaretsang.
Allergie
Ea lintho tse kulang - ho hlaha ha lekhopho letlalong, ho hlohlona.
Tšusumetso ho bokhoni ba taolo ea methapo
Moriana o khona ho ama tlhokomelo e mpe. Ka hona, kalafo ea ho khanna koloi kapa ho sebetsa ka lisebelisoa tse thata ha e khothalletsoe. Bakuli ba lokela ho ba hlokolosi lefifing.
Litaelo tse khethehileng
Sebelisa nakong ea bokhachane le pelehi
Ha ho na boiphihlelo le Aprovel ntlheng ena. Ho ka etsahala lefu la fetal. Ha ho fumanoa bokhachane, lithethefatsi li hlakotsoe ka botlalo.
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Nakong ea ho anyesa, kalafo ea Aprovel e thibetsoe. Haeba ho sa khonehe ho hlakola moriana, o hloka ho fetisetsa lesea ho fepa ka maiketsetso.
Khetho ea Aprovel ho bana ba 300
E thibetsoe, incl. ha a le lilemo li 6.
Sebelisa botsofaling
Ha ho na lebaka la ho fetola litekanyetso tsa moriana ho batho ba tsofetseng.
Kopo ea ts'ebetso ea renal e senyehileng
Haeba mokuli a rerile ho ts'oasa liphekolo, a ka lebelloa ho fokolisa tšebetso ea setho. Sena ke 'nete haholo ho bakuli ba nang le renal artery stenosis. Ho bakuli ba bang, ho ile ha bonoa keketseho ea bongata ba uric acid maling.
Batho ba nang le bothata ba ho hloleha ha menoana ba hloka ho lekola palo ea potasium maling a bona. Ha ho na tlhahisoleseling mabapi le mamello ea lithethefatsi ke bakuli ba nang le phetisetso ea liphio.
Sebelisa bakeng sa ts'ebetso ea sebete e sa sebetseng
Ho hlokahala hore u be hlokolosi ha u sebelisa moriana.
Bongata bo fetang Aprovel 300
Ts'ebeliso ea 900 mg ea Aprovel bakeng sa likhoeli tse peli ha e bake chefo. Ha ho na bopaki ba boteng ba kokoanahloko kalafong.
Bakuli ba nkang ntho e ngata ba hloka ho hlatsoa mala a bona, ho baka ho hlatsa. Hemodialysis ha e na thuso ebile ha ea nepahala.
Ho sebelisana le lithethefatsi tse ling
Ha hoa lumelloa ho sebelisa meriana eohle e nang le aliskiren. Sena se sebetsa ho batho ba nang le lefu la tsoekere le lefu le matla la liphio. Ha e khothalletsoe ho kopanya le li-inhibitors tsa ACE.
Ha u nka meriana ea lithium, ho ka khoneha hore ho be le keketseho ea se kahare sa ntho ena ho plasma.
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Tšebeliso e tšoanang ea Aprovel le lithethefatsi tse ling tsa antihypertgency li ka fokotsa khatello haholo ho fihlela bothateng ba hypotonic. Ts'ebeliso ea li-diuretics ka tekanyetso e phahameng e tlatsetsa ho hypovolemia.
Tekanyo ea joala
Nakong ea kalafo, ho thibetsoe ka thata ho noa joala.
Li-analog
Lifekthering, lithethefatsi lia rekisoa - li-analogues tsa Aprovel. Tsena li kenyeletsa:
- Irbesso;
- Irbetan;
- Istar;
- Converium;
- Rotazar;
- Firmast;
- Ira Sanovel;
- Moemeli;
- Cantab;
- Heathart;
- Angizar
- Lozap.
Lithethefatsi tsa Russia tse nang le phello e ts'oanang - Linsia, Diocor.
Lipehelo tsa khefu ea khemisi
Aprovel e fumaneha litlhare tsa litlama-tlama feela ka lengolo la ngaka.
Theko ea Aprovel 300
Litsenyehelo tsa matlapa a 28 ke li-ruble tse 820.
Maemo a polokelo ea moriana
Boloka sebakeng se lefifi, se pholileng mme o hole le bana.
Letsatsi la ho felloa ke nako
E loketse likhoeli tse 36. Se ke oa sebelisa kamora nako ena.
Moqapi
E hlahisitsoe ke Setsi sa Sanofi Winthrop, 1 rue de la Vierge, Ambares e Lagrave F-33565, Carbon Blanc Cedex, France.
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Bathong ba morabe oa Negroid, phello ea lithethefatsi Aprovel 300 ha e phatlalatsoe.
Litlhahlobo tsa Aprovel 300
Litsebi tsa kelello
Irina, ea lilemo li 45, ngaka ea methapo ea pelo, Moscow: "Ho phalla ha bakuli ba nang le ts'ebetso ea pelo e sa sebetseng le khatello e phahameng ea mali ho ntse ho eketseha ka linako tsohle. Joalo ka kalafo e rarahaneng, ke ba fa moriana o nang le litekanyetso tsa pele tsa 150 mg, mme haeba ho sa lekane, 300 mg. "Ba mamella moriana hantle mme ha ba bue ka litla-morao. Tšusumetso e tla kapele ka ho lekana mme e nka nako e telele."
Stepan, ea lilemo li 48, ngaka ea pelo, Samara. "Bakeng sa bakuli ba nang le khatello ea methapo ea methapo e sa khaotseng, ke fana ka moriana ka lethal dose ea 300 mg hang ka letsatsi, hoseng. Phokotso e boletsoeng ea hore khatello ea mali e shejoa kamora beke bekeng ea kalafo qalong. Haeba u latela lijo, u ka boloka maemo a ho ba 130/80 mm, ka linako tse ling le tlase. Ke khothaletsa thupelo e telele ea tlhokomelo. kalafo (lethal dose e felisitsoe). Sena se ka fokotsa kotsi ea lefu la atherosclerosis. "
Bakuli
Svetlana, ea lilemo li 40, Saratov o re: "Ho opeloa ke hlooho ka nako e telele, ho tepella le ho teneha ho nqobelletse ho bona ngaka, o ile a nthomela ho ngaka ea lefu la pelo. Kamora tlhahlobo, o ile a re Aprovel ea 300 mg. Ha ke utloe matla a eona hanghang: khatello e ile ea fokotseha butle kamora matsatsi a 3. Empa kamora beke kamora hore ke qale ho nwa lipilisi, ka bona boleng ba 125/80 ho tonometer. Ke tlatselletsa kalafo ka lijo le ho noa tee ea litlama. "
Igor, ea lilemo li 58, St. Petersburg: "Ke nka 150 mg ea Aprovel hanngoe ka letsatsi ho thibela khatello ea mali le lefu la pelo. Hammoho le Aspirin Cardio, nka boloka khatello ea ka ea mali e tsitsitse ka nako ea 120 / 75. Ke boetse ke noha li-decoctions tsa semela bakeng sa thibelo e thusang ho loana. sithabela 'me u hloekise methapo ea mali. "
Lidia, ea lilemo li 45, Moscow: "Haufinyane ho bile le koluoa ea khatello ea mali - khatello e ile ea nyoloha ka potlako ho 185/110. Letsatsing le hlahlamang, kamora ho fokotsa khatello, ke ile ka etela ngaka ea lelapa e ileng ea nkeletsa hore ke nke Aprovel 300 mg hoseng ho hong le ho hong. "khatello e phahameng ea mali ha e sa hlola e nkhathatsa. Kamora hore ke qete ho etsa kalafo ea antihypertgency, ke noa lintho tse thusang ho thibela ho nyehlisa."